Diastereoselective construction of anti-4,5-disubstituted-1,3-dioxolanes via a bismuth-mediated two-component hemiacetal oxa-conjugate addition of γ-hydroxy-α,β-unsaturated ketones with paraformaldehyde.

نویسندگان

  • Aleksandr Grisin
  • Samuel Oliver
  • Michael D Ganton
  • John Bacsa
  • P Andrew Evans
چکیده

The bismuth-mediated two-component hemiacetal oxa-conjugate addition of γ-hydroxy-α,β-unsaturated ketones with paraformaldehyde affords anti-4,5-disubstituted-1,3-dioxolanes in an efficient and stereoselective manner. The reaction provides a practical, inexpensive and atom-economical approach to these types of heterocycles, which represent useful intermediates for target-directed synthesis and precursors to syn-1,2-diols.

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عنوان ژورنال:
  • Chemical communications

دوره 51 86  شماره 

صفحات  -

تاریخ انتشار 2015